Literature DB >> 11087559

Design, radiosynthesis, and biodistribution of a new potent and selective ligand for in vivo imaging of the adenosine A(2A) receptor system using positron emission tomography.

S Todde1, R M Moresco, P Simonelli, P G Baraldi, B Cacciari, G Spalluto, K Varani, A Monopoli, M Matarrese, A Carpinelli, F Magni, M G Kienle, F Fazio.   

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Year:  2000        PMID： 11087559     DOI： 10.1021/jm0009843

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  32 in total

Review 1.  Recent developments in adenosine receptor ligands and their potential as novel drugs.

Authors:  Christa E Müller; Kenneth A Jacobson
Journal:  Biochim Biophys Acta       Date:  2010-12-23

2.  Molecular probes for the A2A adenosine receptor based on a pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine scaffold.

Authors:  T Santhosh Kumar; Shilpi Mishra; Francesca Deflorian; Lena S Yoo; Khai Phan; Miklos Kecskés; Angela Szabo; Bidhan Shinkre; Zhan-Guo Gao; William Trenkle; Kenneth A Jacobson
Journal:  Bioorg Med Chem Lett       Date:  2010-11-21       Impact factor: 2.823

Review 3.  Adenosine A2A receptors and basal ganglia physiology.

Authors:  S N Schiffmann; G Fisone; R Moresco; R A Cunha; S Ferré
Journal:  Prog Neurobiol       Date:  2007-06-26       Impact factor: 11.685

4.  Remote control of movement disorders using a photoactive adenosine A2A receptor antagonist.

Authors:  Jaume Taura; Ernest G Nolen; Gisela Cabré; Jordi Hernando; Lucia Squarcialupi; Marc López-Cano; Kenneth A Jacobson; Víctor Fernández-Dueñas; Francisco Ciruela
Journal:  J Control Release       Date:  2018-05-31       Impact factor: 9.776

5.  The Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptors.

Authors:  Stephen P H Alexander; Helen E Benson; Elena Faccenda; Adam J Pawson; Joanna L Sharman; Michael Spedding; John A Peters; Anthony J Harmar
Journal:  Br J Pharmacol       Date:  2013-12       Impact factor: 8.739

6.  Photoaffinity Labeling of the Human A2A Adenosine Receptor and Cross-link Position Analysis by Mass Spectrometry.

Authors:  Hideyuki Muranaka; Takaki Momose; Chiaki Handa; Tomonaga Ozawa
Journal:  ACS Med Chem Lett       Date:  2017-05-17       Impact factor: 4.345

7.  Activation of adenosine A2A or A2B receptors causes hypothermia in mice.

Authors:  Jesse Lea Carlin; Shalini Jain; Romain Duroux; R Rama Suresh; Cuiying Xiao; John A Auchampach; Kenneth A Jacobson; Oksana Gavrilova; Marc L Reitman
Journal:  Neuropharmacology       Date:  2018-03-13       Impact factor: 5.250

8.  Isothermal chemical denaturation to determine binding affinity of small molecules to G-protein coupled receptors.

Authors:  Patrick Ross; Wilhelm Weihofen; Fai Siu; Amy Xie; Hetal Katakia; S Kirk Wright; Ian Hunt; Richard K Brown; Ernesto Freire
Journal:  Anal Biochem       Date:  2014-12-04       Impact factor: 3.365

9.  The adenosine A2A receptor antagonist ZM241385 enhances neuronal survival after oxygen-glucose deprivation in rat CA1 hippocampal slices.

Authors:  A M Pugliese; C Traini; S Cipriani; M Gianfriddo; T Mello; M G Giovannini; A Galli; F Pedata
Journal:  Br J Pharmacol       Date:  2009-05-05       Impact factor: 8.739

10.  Application of the functionalized congener approach to dendrimer-based signaling agents acting through A(2A) adenosine receptors.

Authors:  Yoonkyung Kim; Athena M Klutz; Béatrice Hechler; Zhan-Guo Gao; Christian Gachet; Kenneth A Jacobson
Journal:  Purinergic Signal       Date:  2008-07-04       Impact factor: 3.765
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