Literature DB >> 11052104

Reactivity of 3-iodoimidazo[1,2-a]pyridines using a Suzuki-type cross-coupling reaction.

C Enguehard1, J L Renou, V Collot, M Hervet, S Rault, A Gueiffier.   

Abstract

The influence of base and solvent in Suzuki cross-coupling reaction on various 2-substituted-3-iodoimidazo[1,2-a]pyridines was reported. The reactivity was largely influenced by nature of the substituent. Optimized yields and shortened times of reaction were obtained using strong bases in DME.

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Year:  2000        PMID: 11052104     DOI: 10.1021/jo000698z

Source DB:  PubMed          Journal:  J Org Chem        ISSN: 0022-3263            Impact factor:   4.354


  5 in total

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Authors:  Jiamo Lu; Prabhakar Risbood; Charles T Kane; Md Tafazzal Hossain; Larry Anderson; Kimberly Hill; Anne Monks; Yongzhong Wu; Smitha Antony; Agnes Juhasz; Han Liu; Guojian Jiang; Erik Harris; Krishnendu Roy; Jennifer L Meitzler; Mariam Konaté; James H Doroshow
Journal:  Biochem Pharmacol       Date:  2017-07-11       Impact factor: 5.858

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Authors:  Brendan Frett; Nick McConnell; Catherine C Smith; Yuanxiang Wang; Neil P Shah; Hong-yu Li
Journal:  Eur J Med Chem       Date:  2015-02-28       Impact factor: 6.514

3.  Efficient access to 2,3-diarylimidazo[1,2-a]pyridines via a one-pot, ligand-free, palladium-catalyzed three-component reaction under microwave irradiation.

Authors:  Yuanxiang Wang; Brendan Frett; Hong-yu Li
Journal:  Org Lett       Date:  2014-05-22       Impact factor: 6.005

4.  Metal-free C-H arylation of imidazoheterocycles with aryl hydrazines.

Authors:  Sourav Jana; Sadhanendu Samanta; Avik K Bagdi; Valerii Z Shirinian; Alakananda Hajra
Journal:  RSC Adv       Date:  2018-04-03       Impact factor: 3.361

5.  Regiocontrolled microwave assisted bifunctionalization of 7,8-dihalogenated imidazo[1,2-a]pyridines: a one pot double-coupling approach.

Authors:  Emilie Marie; Sébastien Bouclé; Cécile Enguehard-Gueiffier; Alain Gueiffier
Journal:  Molecules       Date:  2012-09-06       Impact factor: 4.411

  5 in total

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