Literature DB >> 10983288

1,5-benzodiazepine derivatives of 3-arylsydnones: synthesis and antimicrobial activity of 3-aryl-4-[2'-aryl-2',4',6',7'-tetrahydro-(1'H)-1',5'-benzodiazepine-4' -yl]sydnones.

J R Kavali1, B V Badami.   

Abstract

The alpha-beta-unsaturated ketones of 3-arylsydnones (Ia-y) were treated with 1,2-phenylenediamine to obtain the 3-aryl-4-[2'-aryl- 2',4',6',7'-tetrahydro-(1'H)-1',5'-benzodiazepine-4'-yl]sydnones (IIa-y) in high yield. All the new compounds synthesised were screened for antibacterial and antifungal activities.

Entities:  

Mesh：

Substances：

Year:  2000        PMID： 10983288     DOI： 10.1016/s0014-827x(00)00061-6

Source DB:  PubMed          Journal:  Farmaco        ISSN： 0014-827X


  3 in total

1.  A facile synthesis and antimicrobial activity evaluation of sydnonyl-substituted thiazolidine derivatives.

Authors:  Mei-Hsiu Shih; Yu-Yuan Xu; Yu-Sheng Yang; Guan-Ling Lin
Journal:  Molecules       Date:  2015-04-13       Impact factor: 4.411

2.  Synthesis and catalytic evaluation of PVP-CeO2/rGO as a highly efficient and recyclable heterogeneous catalyst for multicomponent reactions in water.

Authors:  Shaheen Siddiqui; Zeba N Siddiqui
Journal:  Nanoscale Adv       Date:  2020-08-28

3.  Synthesis and antibacterial and antifungal activities of N-(tetra-O-acetyl-β-d-glucopyranosyl)thiosemicarbazones of substituted 4-formylsydnones.

Authors:  Nguyen Dinh Thanh; Hoang Thanh Duc; Vu Thi Duyen; Phan Manh Tuong; Nguyen Van Quoc
Journal:  Chem Cent J       Date:  2015-10-19       Impact factor: 4.215
  3 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.