Literature DB >> 10888320

Syntheses and antifilarial profile of 7-chloro-4-(substituted amino) quinolines: a new class of antifilarial agents.

S Tewari1, P M Chauhan, A P Bhaduri, N Fatima, R K Chatterjee.   

Abstract

The syntheses of 7-chloro-4-(substituted amino) quinolines (2-22) and their antifilarial activities are delineated. Some of the screened compounds have shown promising filarial response and sterilization effect on female Acanthocheilonema viteae in rodents.

Entities:  

Mesh：

Substances：

Year:  2000        PMID： 10888320     DOI： 10.1016/s0960-894x(00)00255-9

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  4 in total

1.  In vitro antifilarial activity of glutathione S-transferase inhibitors.

Authors:  Lakshmy Srinivasan; Nisha Mathew; Kalyanasundaram Muthuswamy
Journal:  Parasitol Res       Date:  2009-06-28       Impact factor: 2.289

2.  A controlled trial to assess the effect of quinine, chloroquine, amodiaquine, and artesunate on Loa loa microfilaremia.

Authors:  Joseph Kamgno; Patrick Nguipdop Djomo; Sébastien D Pion; Björn Thylefors; Michel Boussinesq
Journal:  Am J Trop Med Hyg       Date:  2010-03       Impact factor: 2.345

3.  Modular Three-Component Synthesis of 4-Aminoquinolines via an Imidoylative Sonogashira/Cyclization Cascade.

Authors:  Jurriën W Collet; Kelly Ackermans; Jeffrey Lambregts; Bert U W Maes; Romano V A Orru; Eelco Ruijter
Journal:  J Org Chem       Date:  2018-01-02       Impact factor: 4.354

4.  Antifilarial lead molecules isolated from Trachyspermum ammi.

Authors:  Nisha Mathew; Shailja Misra-Bhattacharya; Vanamail Perumal; Kalyanasundaram Muthuswamy
Journal:  Molecules       Date:  2008-09-11       Impact factor: 4.411
  4 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.