Literature DB >> 10767039

Discovery of Carbohydrate Sulfotransferase Inhibitors from a Kinase-Directed Library We thank Sharon Long and Dave Keating for providing both the NodH sulfotransferase and APS Kinase during our preliminary experiments and Jack Kirsch for numerous helpful conversations. J.I.A. and K.G.B were supported by NIH Molecular Biophysics Training Grant (No. T32GM0895). This research was funded by grants to C.R.B. from the Pew Scholars Program, the W. M. Keck Foundation and the American Cancer Society (Grant No. RPG9700501BE).

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Abstract

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Year:  2000        PMID: 10767039     DOI: 10.1002/(sici)1521-3773(20000403)39:7<1303::aid-anie1303>3.0.co;2-0

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN: 1433-7851            Impact factor:   15.336


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  12 in total

1.  Mass spectrometry and immobilized enzymes for the screening of inhibitor libraries.

Authors:  M T Cancilla; M D Leavell; J Chow; J A Leary
Journal:  Proc Natl Acad Sci U S A       Date:  2000-10-24       Impact factor: 11.205

Review 2.  New targets and inhibitors of mycobacterial sulfur metabolism.

Authors:  Hanumantharao Paritala; Kate S Carroll
Journal:  Infect Disord Drug Targets       Date:  2013-04

Review 3.  Modifications of glycans: biological significance and therapeutic opportunities.

Authors:  Saddam M Muthana; Christopher T Campbell; Jeffrey C Gildersleeve
Journal:  ACS Chem Biol       Date:  2012-01-11       Impact factor: 5.100

Review 4.  Recent advances in sulfotransferase enzyme activity assays.

Authors:  Priscilla Paul; Jiraporn Suwan; Jian Liu; Jonathan S Dordick; Robert J Linhardt
Journal:  Anal Bioanal Chem       Date:  2012-04-12       Impact factor: 4.142

5.  Inhibitory peptides of the sulfotransferase domain of the heparan sulfate enzyme, N-deacetylase-N-sulfotransferase-1.

Authors:  Tarsis F Gesteira; Vivien J Coulson-Thomas; Alessandro Taunay-Rodrigues; Vitor Oliveira; Bryan E Thacker; Maria A Juliano; Renata Pasqualini; Wadih Arap; Ivarne L S Tersariol; Helena B Nader; Jeffrey D Esko; Maria A S Pinhal
Journal:  J Biol Chem       Date:  2010-02-02       Impact factor: 5.157

Review 6.  Drug targets in mycobacterial sulfur metabolism.

Authors:  Devayani P Bhave; Wilson B Muse; Kate S Carroll
Journal:  Infect Disord Drug Targets       Date:  2007-06

7.  A structural and biochemical basis for PAPS-independent sulfuryl transfer by aryl sulfotransferase from uropathogenic Escherichia coli.

Authors:  Goran Malojcić; Robin L Owen; John P A Grimshaw; Maurice S Brozzo; Hiang Dreher-Teo; Rudi Glockshuber
Journal:  Proc Natl Acad Sci U S A       Date:  2008-11-26       Impact factor: 11.205

8.  Small-molecule inhibition of pyruvate phosphate dikinase targeting the nucleotide binding site.

Authors:  Alexander Minges; Georg Groth
Journal:  PLoS One       Date:  2017-07-10       Impact factor: 3.240

Review 9.  The Regulation of Steroid Action by Sulfation and Desulfation.

Authors:  Jonathan W Mueller; Lorna C Gilligan; Jan Idkowiak; Wiebke Arlt; Paul A Foster
Journal:  Endocr Rev       Date:  2015-07-27       Impact factor: 19.871

10.  New tools for carbohydrate sulfation analysis: heparan sulfate 2-O-sulfotransferase (HS2ST) is a target for small-molecule protein kinase inhibitors.

Authors:  Dominic P Byrne; Yong Li; Krithika Ramakrishnan; Igor L Barsukov; Edwin A Yates; Claire E Eyers; Dulcé Papy-Garcia; Sandrine Chantepie; Vijayakanth Pagadala; Jian Liu; Carrow Wells; David H Drewry; William J Zuercher; Neil G Berry; David G Fernig; Patrick A Eyers
Journal:  Biochem J       Date:  2018-08-14       Impact factor: 3.857

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