Literature DB >> 10673087

Solution-phase combinatorial synthesis and evaluation of piperazine-2,5-dione derivatives.

W A Loughlin1, R L Marshall, A Carreiro, K E Elson.   

Abstract

An efficient one-pot synthesis of a 61-membered combinatorial chemistry library of piperazine-2,5-diones was accomplished. Results of combinatorial synthesis, purification, analysis, and biological evaluation are described.

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Year:  2000        PMID： 10673087     DOI： 10.1016/s0960-894x(99)00634-4

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  5 in total

Review 1.  Exploring privileged structures: the combinatorial synthesis of cyclic peptides.

Authors:  Douglas A Horton; Gregory T Bourne; Mark L Smythe
Journal:  J Comput Aided Mol Des       Date:  2002 May-Jun       Impact factor: 3.686

Review 2.  Exploring privileged structures: the combinatorial synthesis of cyclic peptides.

Authors:  Douglas A Horton; Gregory T Bourne; Mark L Smythe
Journal:  Mol Divers       Date:  2002       Impact factor: 2.943

3.  Solid-phase total synthesis of (-)-Phenylhistine and (-)-Aurantiamine. Synthesis of a diverse dehydro-2,5-diketopiperazine library. Part II.

Authors:  Elias A Couladouros; Alexandros D Magos
Journal:  Mol Divers       Date:  2005       Impact factor: 2.943

4.  Microwave-assisted solution-phase synthesis and DART-mass spectrometric monitoring of a combinatorial library of indolin-2,3-dione schiff bases with potential antimycobacterial activity.

Authors:  Tarek Aboul-Fadl; Hatem A Abdel-Aziz; Adnan Kadi; Pervez Ahmad; Tilal Elsaman; Mohamed W Attwa; Ibrahim A Darwish
Journal:  Molecules       Date:  2011-06-22       Impact factor: 4.411

Review 5.  Cyclic Dipeptides: The Biological and Structural Landscape with Special Focus on the Anti-Cancer Proline-Based Scaffold.

Authors:  Joanna Bojarska; Adam Mieczkowski; Zyta M Ziora; Mariusz Skwarczynski; Istvan Toth; Ahmed O Shalash; Keykavous Parang; Shaima A El-Mowafi; Eman H M Mohammed; Sherif Elnagdy; Maha AlKhazindar; Wojciech M Wolf
Journal:  Biomolecules       Date:  2021-10-14
  5 in total

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