Literature DB >> 10458808

A One-Pot, One-Operation

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Abstract

Enantiomerically pure 2,1-benzothiazines are readily prepared by a one-pot, one-operation procedure consisting of a palladium-catalyzed aryl amination of an ortho-bromobenzaldehyde with a sulfoximine followed by an intramolecular condensation reaction [Eq. (1)]. BINAP=1,1'-binaphthalene-2,2'-diylbis(diphenylphosphane).

Entities:  

Year:  1999        PMID： 10458808     DOI： 10.1002/(sici)1521-3773(19990816)38:16<2419::aid-anie2419>3.0.co;2-i

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


  10 in total

1.  Toward the total synthesis of elisapterosin B: A Hg(OTf)(2)-promoted diastereoselective intramolecular Friedel-Crafts alkylation reaction.

Authors:  Weijiang Ying; Charles L Barnes; Michael Harmata
Journal:  Tetrahedron Lett       Date:  2011-01-12       Impact factor: 2.415

2.  Preparation of S-2-halophenyl-2,1-benzothiazines.

Authors:  Aswin Garimalla; Michael Harmata
Journal:  Tetrahedron       Date:  2021-02-10       Impact factor: 2.457

Review 3.  Synthesis and Transformations of NH-Sulfoximines.

Authors:  Michael Andresini; Arianna Tota; Leonardo Degennaro; James A Bull; Renzo Luisi
Journal:  Chemistry       Date:  2021-10-13       Impact factor: 5.020

4.  Benzothiazines in synthesis. Further studies of the intramolecular, stereoselective addition of sulfonimidoyl carbanions to alpha,beta-unsaturated functional groups.

Authors:  Michael Harmata; Kanok-on Rayanil; Vinson R Espejo; Charles L Barnes
Journal:  J Org Chem       Date:  2009-04-17       Impact factor: 4.354

5.  Benzothiazines in synthesis. A formal total synthesis of pseudopteroxazole.

Authors:  Michael Harmata; Zhengxin Cai; Yugang Chen
Journal:  J Org Chem       Date:  2009-08-07       Impact factor: 4.354

6.  Novel Pieces for the Emerging Picture of Sulfoximines in Drug Discovery: Synthesis and Evaluation of Sulfoximine Analogues of Marketed Drugs and Advanced Clinical Candidates.

Authors:  Juan Alberto Sirvent; Ulrich Lücking
Journal:  ChemMedChem       Date:  2017-03-22       Impact factor: 3.466

7.  N-Arylation of NH-Sulfoximines via Dual Nickel Photocatalysis.

Authors:  Alexander Wimmer; Burkhard König
Journal:  Org Lett       Date:  2019-04-02       Impact factor: 6.005

8.  Modern Stereoselective Synthesis of Chiral Sulfinyl Compounds.

Authors:  Elżbieta Wojaczyńska; Jacek Wojaczyński
Journal:  Chem Rev       Date:  2020-04-29       Impact factor: 60.622

9.  Identification of Atuveciclib (BAY 1143572), the First Highly Selective, Clinical PTEFb/CDK9 Inhibitor for the Treatment of Cancer.

Authors:  Ulrich Lücking; Arne Scholz; Philip Lienau; Gerhard Siemeister; Dirk Kosemund; Rolf Bohlmann; Hans Briem; Ildiko Terebesi; Kirstin Meyer; Katja Prelle; Karsten Denner; Ulf Bömer; Martina Schäfer; Knut Eis; Ray Valencia; Stuart Ince; Franz von Nussbaum; Dominik Mumberg; Karl Ziegelbauer; Bert Klebl; Axel Choidas; Peter Nussbaumer; Matthias Baumann; Carsten Schultz-Fademrecht; Gerd Rühter; Jan Eickhoff; Michael Brands
Journal:  ChemMedChem       Date:  2017-10-16       Impact factor: 3.466

10.  Visible-Light-Mediated Photoredox-Catalyzed N-Arylation of NH-Sulfoximines with Electron-Rich Arenes.

Authors:  Alexander Wimmer; Burkhard König
Journal:  Adv Synth Catal       Date:  2018-08-02       Impact factor: 5.837
  10 in total

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