Literature DB >> 10230641

Use of the Suzuki reaction for the synthesis of aryl-substituted heterocycles as corticotropin-releasing hormone (CRH) antagonists.

A J Cocuzza1, D R Chidester, S Culp, L Fitzgerald, P Gilligan.   

Abstract

The Suzuki reaction has been used to synthesize a variety of aryl-substituted heterocyclic antagonists of the CRH1 receptor. Examples with several different heterocyclic cores are potent CRH receptor ligands.

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Year:  1999        PMID: 10230641     DOI: 10.1016/s0960-894x(99)00133-x

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN: 0960-894X            Impact factor:   2.823


  3 in total

Review 1.  Recent advances in the application of indoles in multicomponent reactions.

Authors:  Ghodsi Mohammadi Ziarani; Razieh Moradi; Tahereh Ahmadi; Negar Lashgari
Journal:  RSC Adv       Date:  2018-03-28       Impact factor: 4.036

2.  Synthesis, characterization and in vitro anti-tumor activities of novel 9-ethyl-9H-purine derivatives.

Authors:  Raghu Ningegowda; Amit Grover; S Ranjith; Kanchugarakoppal S Rangappa; B S Priya; S Nanjunda Swamy
Journal:  Invest New Drugs       Date:  2009-09-16       Impact factor: 3.850

3.  Visible-Light-Induced C-C Coupling Reaction to Synthesize Bipyridine From 3-Cyano-1,4-Dihydropyridines.

Authors:  Shijun Chen; Qidi Zhong; Hao Zhu; Chunyan Liu; Pengyu Zhuang; Wuji Sun
Journal:  Front Chem       Date:  2020-01-17       Impact factor: 5.221

  3 in total

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